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Book:

1. Masahiro Yoshida and Yoshimitsu Nagao :
Transition metal-catalyzed ring expansion cyclization reactions,
Wiley-VCH, Weinheim, Nov. 2009.
2. Yoshimitsu Nagao and Shigeki Sano :
Electronic Encyclopedia of Reagents for Organic Synthesis, --- (S)-4-Isopropyl-1,3-thiazolidine-2-thione ---,
John Wiley & Sons, Inc., Chichester, 2008.
3. Malcolm Sainsbury, Yoshimitsu Nagao and Shigeki Sano :
Tutorial Chemistry Texts 7, --- Heterocyclic Chemistry ---,
Kagaku-Dojin Publishing Company,INC, Kyoto, Oct. 2004.
4. Hirofumi Shibata and Yoshimitsu Nagao :
メディシナルケミストリー,
MARUZEN Co.,Ltd., Tokyo, Mar. 2003.
5. Yoshimitsu Nagao and Shigeki Sano :
創薬化学の基礎となる不斉反応1,
株式会社 廣川書店, Tokyo, Feb. 1998.

Academic Paper (Judged Full Paper):

1. Shigeki Sano, Takashi Ichikawa, Michiyasu Nakao and Yoshimitsu Nagao :
Deconjugative Esterification of 2-(4-Phenylcyclohexylidne)acetic Acid via Intramolecular Chirality Transfer,
Chemistry Letters, Vol.41, No.2, 189-190, 2012.
(DOI: 10.1246/cl.2012.189,   CiNii: 1360846644041797248)
2. Shigeki Sano, Takashi Ichikawa, Michiyasu Nakao and Yoshimitsu Nagao :
A Microwave-Assisted Deconjugative Esterification of α,β-Unsaturated Carboxylic Acids through alpha,beta-Unsaturated Ketene Intermediates,
Chemistry Letters, Vol.41, No.1, 68-69, 2012.
(DOI: 10.1246/cl.2012.68)
3. Shigeki Sano, Yoshinori Okubo, Atsushi Handa, Michiyasu Nakao, Syuji Kitaike, Yoshimitsu Nagao and Hisao Kakegawa :
Reinvestigation of the Synthesis of Isoliquiritigenin (ILG): Application of Horner-Wadsworth-Emmons Reaction and Claisen-Schmidt Condensation,
Chemical & Pharmaceutical Bulletin, Vol.59, No.7, 885-888, 2011.
(DOI: 10.1248/cpb.59.885,   PubMed: 21720042)
4. Shigeki Sano, Takeshi Tsumura, Noriaki Tanimoto, Takashi Honjo, Michiyasu Nakao and Yoshimitsu Nagao :
Modified Cinchona Alkaloid-Zinc Complex Catalysts: Enantioselective Monoacetylation of Glycerol Derivatives with Acetic Anhydride,
Synlett, No.2, 256-260, 2010.
(DOI: 10.1055/s-0029-1218562)
5. Takashi Honjo, Takeshi Tsumura, Shigeki Sano, Yoshimitsu Nagao, Kentaro Yamaguchi and Yoshihisa Sei :
A Chiral Bifunctional Sulfonamide as an Organocatalyst: Alcoholysis of -Symmetric Cyclic Dicarboxylic Anhydrides,
Synlett, No.20, 3279-3282, 2009.
(DOI: 10.1055/s-0029-1218374)
6. Kazuhiko Hayashi, Eiko Kujime, Hajime Katayama, Shigeki Sano, Motoo Shiro and Yoshimitsu Nagao :
Synthesis and Reaction of 1-Azabicyclo[3.1.0]hexane,
Chemical & Pharmaceutical Bulletin, Vol.57, No.10, 1142-1146, 2009.
(DOI: 10.1248/cpb.57.1142,   PubMed: 19801877)
7. Kazuhiko Hayashi, Eiko Kujime, Hajime Katayama, Shigeki Sano and Yoshimitsu Nagao :
Reaction of 1-Azabicyclo[1.1.0]butane with Activated Amides,
Heterocycles, Vol.78, No.1, 1777-1786, 2009.
(DOI: 10.3987/COM-09-11677,   CiNii: 1521136280100788864)
8. Shigeki Sano, Michiyasu Nakao, Masanori Takeyasu, Syuji Kitaike, Yasuko Yoshioka and Yoshimitsu Nagao :
Use of Diketopiperazines for Determining Absolute Configurations of α-Substituted Serines by 1H-NMR Spectroscopy,
Heterocycles, Vol.79, No.1, 781-789, 2009.
(DOI: 10.3987/COM-08-S(D)47,   CiNii: 1520010379846386176)
9. Shigeki Sano, Michiyasu Nakao, Masanori Takeyasu, Chiyo Yamamoto, Syuji Kitaike, Yasuko Yoshioka and Yoshimitsu Nagao :
Chemoenzymatic Synthesis of α-Substituted Serines via Enantiodivergent Transformation,
The Open Organic Chemistry Journal, Vol.3, 22-34, 2009.
(DOI: 10.2174/1874095200903010022)
10. Kazuhiko Hayazhi, Shiho Ogawa, Shigeki Sano, Motoo Shiro, Kentaro Yamaguchi, Yoshihisa Sei and Yoshimitsu Nagao :
Intramolecular Nonbonded S---N Interaction in Rabeprazole,
Chemical & Pharmaceutical Bulletin, Vol.56, No.6, 802-806, 2008.
(DOI: 10.1248/cpb.56.802,   PubMed: 18520084,   CiNii: 1390001204170061568)
11. Yoshifumi Ikee, Kana Hashimoto, Mai Kamino, Masaaki Nakashima, Kazuhiko Hayazhi, Shigeki Sano, Motoo Shiro and Yoshimitsu Nagao :
Synthesis of New Quinolone Antibiotics Utilizing Azetidine Derivatives Obtained from 1-Azabicyclo[1.1.0]butane,
Chemical & Pharmaceutical Bulletin, Vol.56, No.3, 346-356, 2008.
(DOI: 10.1248/cpb.56.346,   PubMed: 18310947,   CiNii: 1390001204168894336)
12. Kazuhiko Hayashi, Eiko Kujime, Hajime Katayama, Shigeki Sano and Yoshimitsu Nagao :
Effects of Magnesium Salts and Amines on the Stereoselectivity in the Imine Aldol Reaction,
Chemical & Pharmaceutical Bulletin, Vol.55, No.12, 1773-1775, 2007.
(DOI: 10.1248/cpb.55.1773,   PubMed: 18057758,   CiNii: 1390001204168630016)
13. Takashi Honjo, Michiyasu Nakao, Shigeki Sano, Motoo Shiro, Kentaro Yamaguchi, Yoshihisa Sei and Yoshimitsu Nagao :
Nonenzymatic Enantioselective Monoacetylation of Prochiral 2-Protectedamino-2-alkyl-1,3-propanediols Utilizing a Chiral Sulfonamide-Zn Complex Catalyst,
Organic Letters, Vol.9, No.3, 509-512, 2007.
(DOI: 10.1021/ol063063g,   PubMed: 17249799)
14. Chung Keun Jin, Toshiaki Yamada, Shigeki Sano, Motoo Shiro and Yoshimitsu Nagao :
Stereoselective Synthesis of Unsymmetrical Conjugated Dienes and Trienes Utilizing Silacyclobutenes,
Tetrahedron Letters, Vol.48, No.21, 3671-3675, 2007.
(DOI: 10.1016/j.tetlet.2007.03.122)
15. Yoshifumi Ikee, Kana Hashimoto, Masaaki Nakashima, Kazuhiko Hayashi, Shigeki Sano, Motoo Shiro and Yoshimitsu Nagao :
Synthesis and Antibacterial Activities of New Quinolone Derivatives Utilizing 1-Azabicyclo[1.1.0]butane,
Bioorganic & Medicinal Chemistry Letters, Vol.17, No.4, 942-945, 2007.
(DOI: 10.1016/j.bmcl.2006.11.048,   PubMed: 17157008)
16. Chung Keun Jin, Tinh Van Dang, Yoshifumi Ikee, Toshiaki Yamada, Shigeki Sano, Motoo Shiro and Yoshimitsu Nagao :
Synthesis of Novel Silacyclobutene Derivatives Utilizing Zirconocene- and Titanocene-ethylene Complexes,
Heterocycles, Vol.70, No.1, 71-75, 2006.
(CiNii: 1523388079969080832,   Elsevier: Scopus)
17. Shigeki Sano, Yoko Kuroda, Katsuyuki Saito, Yukiko Ose and Yoshimitsu Nagao :
Tandem Reduction Olefination of Triethyl 2-Aceyl-2-fluoro-2-phosphonoacetates and a Synthetic Approach to Cbz-Gly-Ψ[(Z)-CF=C]-Gly Dipeptide Isostere,
Tetrahedron, Vol.62, No.51, 11881-11890, 2006.
(DOI: 10.1016/j.tet.2006.09.096,   Elsevier: Scopus)
18. Shigeki Sano, Etsuko Harada, Tomohiro Azetsu, Takashi Ichikawa, Michiyasu Nakao and Yoshimitsu Nagao :
Novel Deconjugative Esterification of 2-Cyclohexylidneacetic Acids through 4-(Pyrrolidin-1-yl)pyridine Catalyzed Carbodiimide Couplings,
Chemistry Letters, Vol.35, No.11, 1286-1287, 2006.
(DOI: 10.1246/cl.2006.1286,   CiNii: 1360846644040903936)
19. Shigeki Sano, Shinobu Abe, Tomohiro Azetsu, Michiyasu Nakao, Motoo Shiro and Yoshimitsu Nagao :
Diastereoselective Horner-Wadsworth-Emmons Reaction for the Synthesis of Tetrasubstituted Alkenes with an Axis of Chirality,
Letters in Organic Chemistry, Vol.3, No.11, 798-801, 2006.
(DOI: 10.2174/157017806779116969,   Elsevier: Scopus)
20. Tinh Van Dang, Chung Keun Jin, Motoyuki Miyamoto, Yoshifumi Ikee, Takashi Masuda, Shigeki Sano, Motoo Shiro and Yoshimitsu Nagao :
Practical Synthesis of New Chiral cis-Phthalazinones with Potential for High Phosphodiesterase (PDE-4) Inhibitory Activity,
Heterocycles, Vol.68, No.10, 2133-2144, 2006.
(CiNii: 1521699230914034304,   Elsevier: Scopus)
21. Shigeki Sano, Michiyasu Nakao, Masanori Takeyasu, Takashi Honjo and Yoshimitsu Nagao :
Lipase-catalyzed Enantioselective Acetylation of Prochiral N-Cbz-2-Alkyl-2-amino-1,3-propanediols and Enantiodivergent Synthesis of α-Benzylserine,
Letters in Organic Chemistry, Vol.3, No.10, 764-767, 2006.
(DOI: 10.2174/157017806779025924,   Elsevier: Scopus)
22. Mihiro Yano, Naoki Muguruma, Susumu Ito, Eriko Aoyagi, Tetsuo Kimura, Yoshitaka Imoto, Jianxin Cao, Shohei Inoue, Shigeki Sano, Yoshimitsu Nagao and Hiroshi Kido :
Fab fragment labeled with ICG-derivative for detecting digestive tract cancer,
Photodiagnosis and Photodynamic Therapy, Vol.3, No.3, 177-183, 2006.
(DOI: 10.1016/j.pdpdt.2006.03.012)
23. Shigeki Sano, Motoyuki Miyamoto, Tomoko Mitani and Yoshimitsu Nagao :
A Novel and Efficient Darzens Reaction Catalyzed by Magnesium Bromide,
Heterocycles, Vol.68, No.3, 459-463, 2006.
(DOI: 10.3987/COM-06-10689,   CiNii: 1522262178384044032,   Elsevier: Scopus)
24. Yoko Tadatsu, Naoki Muguruma, Susumu Ito, Masaya Tadatsu, Yoshihiro Kusaka, Koichi Okamoto, Yoshitaka Imoto, Hiromi Taue, Shigeki Sano and Yoshimitsu Nagao :
Optimal Labeling Condition of Antibodies Available for Immunofluorescence Endoscopy,
The Journal of Medical Investigation : JMI, Vol.53, No.1/2, 52-60, 2006.
(Tokushima University Institutional Repository: 110788,   DOI: 10.2152/jmi.53.52,   PubMed: 16537996)
25. Shigeki Sano, Hisashi Shimizu, Kweon Kim, Woo Song Lee, Motoo Shiro and Yoshimitsu Nagao :
Expeditious Syntheses of Conjugated Allenyl Esters and Oxazoles through a Cascade Reaction of α-Alkynyl Malonates under Alkaline Conditions,
Chemical & Pharmaceutical Bulletin, Vol.54, No.2, 196-203, 2006.
(DOI: 10.1248/cpb.54.196,   PubMed: 16462063,   Elsevier: Scopus)
26. Yoshimitsu Nagao, Satoshi Miyamoto, Motoyuki Miyamoto, Hiroe Takeshige, Kazuhiko Hayashi, Shigeki Sano, Motoo Shiro, Kentaro Yamaguchi and Yoshihisa Sei :
Highly Stereoselective Asymmetric Pummerer Reactions That Incorporate Intermolecular and Intramolecular Nonbonded S---O Interactions,
Journal of the American Chemical Society, Vol.128, No.30, 9722-9729, 2006.
(DOI: 10.1021/ja056649r,   PubMed: 16866527,   Elsevier: Scopus)
27. Takashi Honjo, Shigeki Sano, Motoo Shiro and Yoshimitsu Nagao :
Highly Enantioselective Catalytic Thiolysis of Prochiral Cyclic Dicarboxylic Anhydrides Utilizing a Bifunctional Chiral Sulfonamide,
Angewandte Chemie International Edition, Vol.44, No.36, 5838-5841, 2005.
(DOI: 10.1002/anie.200501408,   PubMed: 16080228)
28. Tinh Van Dang, Motoyuki Miyamoto, Shigeki Sano, Motoo Shiro and Yoshimitsu Nagao :
Practical Synthesis of Chiral cis-Cyclohex-4-ene-1,2-dicarboxylic Acid Derivatives by Utilizing (4S)-Isopropyl-1,3-thiazolidine-2-thione,
Heterocycles, Vol.65, No.5, 1139-1157, 2005.
(DOI: 10.3987/COM-05-10356,   CiNii: 1524232505655234432,   Elsevier: Scopus)
29. Shigeki Sano, Eiko Kujime, Yuka Takemoto, Shiro Motoo and Yoshimitsu Nagao :
A Facile Synthesis of Novel Chiral Phosphonoacetates Bearing a Stereogenic Phosphorus Atom,
Chemical & Pharmaceutical Bulletin, Vol.53, No.1, 131-134, 2005.
(DOI: 10.1248/cpb.53.131,   PubMed: 15635249)
30. Shigeki Sano, Hisashi Shimizu and Yoshimitsu Nagao :
Trimethylaluminum-Induced Diastereoselective Methylation onto Ethyl 2-Oxocyclopentane-1-carboxylate and Isomerization between Both of the Dimethylaluminium-Alkoxide Products,
Tetrahedron Letters, Vol.46, No.16, 2887-2891, 2005.
(DOI: 10.1016/j.tetlet.2005.02.142)
31. Shigeki Sano, Hisashi Shimizu and Yoshimitsu Nagao :
Facile Generation Method for Conjugated Allenyl Esters Based on retro-Dieckmann Type Ring-Opening Reactions,
Tetrahedron Letters, Vol.46, No.16, 2883-2886, 2005.
(DOI: 10.1016/j.tetlet.2005.02.138)
32. Yoshimitsu Nagao, Satoru Tanaka, Akiharu Ueki, Masunori Kumazawa, Satoru GOTO, Takashi Ooi, Shigeki Sano and Motoo Shiro :
New Ring-Expansion Reactions of Hydroxy Propenoyl Cyclic Compounds under Palladium(0)/Phosphine-Catalyzed Conditions,
Organic Letters, Vol.6, No.13, 2133-2136, 2004.
(DOI: 10.1021/ol049450c,   PubMed: 15200303)
33. Yoshimitsu Nagao, Satoru Tanaka, Kazuhiko Hayashi, Shigeki Sano and Motoo Shiro :
New Synthetic Methods for Seven- and Eight-Membered Cyclic Ethers Based on the Ring-Expansion Reactions of Hydroxy or Lithioxy Methoxyallenylisochroman Derivatives,
Synlett, Vol.0, No.3, 481-484, 2004.
(DOI: 10.1055/s-2004-815440,   Elsevier: Scopus)
34. Kazuhiko Hayashi, Yoshifumi Ikee, Satoru GOTO, Motoo Shiro and Yoshimitsu Nagao :
Mechanistic considerations for the consecutive cyclization of 2,3-dibromopropylamine hydrobromide giving a strained molecule, 1-azabicyclo[1.1.0]butane,
Chemical & Pharmaceutical Bulletin, Vol.52, No.1, 89-94, 2004.
(DOI: 10.1248/cpb.52.89,   PubMed: 14709873,   CiNii: 1390001204171270784)
35. Yoshimitsu Nagao, Takashi Honjo, Hitoshi Iimori, Satoru GOTO, Shigeki Sano, Motoo Shiro, Kentaro Yamaguchi and Yoshihisa Sei :
Intramolecular Nonbonded S---O Interaction in Acetazolamide and Thiadiazolinethione Molecules in Their Dimeric Crystalline Structures and Complex Crystalline Structures with Enzymes,
Tetrahedron Letters, Vol.45, No.47, 8757-8761, 2004.
(DOI: 10.1016/j.tetlet.2004.09.103)
36. Masaya Tadatsu, Susumu Ito, Naoki Muguruma, Yoshihiro Kusaka, Kumi Inayama, Termi Bando, Yoko Tadatsu, Koichi Okamoto, Kunio Ii, Yoshimitsu Nagao, Shigeki Sano and Hiromi Taue :
A New Infrared Fluorescent-Labeling Agent and Labeled Antibody for Diagnosing Microcancers,
Bioorganic & Medicinal Chemistry, Vol.11, No.15, 3289-3294, 2003.
(DOI: 10.1016/S0968-0896(03)00239-6,   PubMed: 12837539,   Elsevier: Scopus)
37. Shigeki Sano, Rie Teranishi, Fumihito Nakano, Kyougetu In, Hiroe Takeshige, Takahiro Ishii, Motoo Shiro and Yoshimitsu Nagao :
Asymmetric Horner-Wadsworth-Emmons Reaction Utilizing Isomannide and Isosorbide Derivatives as Chiral Auxiliaries,
Heterocycles, Vol.59, No.2, 793-804, 2003.
(CiNii: 1520291855223705344,   Elsevier: Scopus)
38. Shigeki Sano, Katsuyuki Saito and Yoshimitsu Nagao :
Tandem Reduction-Olefination for the Stereoselective Synthesis of (Z)-α-Fluoro-α,β-unsaturated Esters,
Tetrahedron Letters, Vol.44, No.20, 3987-3990, 2003.
(DOI: 10.1016/S0040-4039(03)00778-0,   CiNii: 1571698601677444480)
39. Shigeki Sano, Yuka Takemoto and Yoshimitsu Nagao :
(E)-Selective Horner Wadsworth Emmons reaction of aldehydes with bis-(2,2,2-trifluoroethyl)phosphonoacetic acid,
ARKIVOC, No.8, 93-101, 2003.
(DOI: 10.3998/ark.5550190.0004.810,   Elsevier: Scopus)
40. Akiharu Ueki, Satoru Tanaka, Masunori Kumazawa, Takashi Ooi, Shigeki Sano and Yoshimitsu Nagao :
A New Convenient Method for Synthesis of 3-(2-Oxoethylidene)isoindolin-1-ones Employing Palladium(II) Acetate and DDQ,
Heterocycles, Vol.61, 449-457, 2003.
(Elsevier: Scopus)
41. Shigeki Sano, Yuka Takemoto and Yoshimitsu Nagao :
(E)-Selective Horner-Wadsworth-Emmons Reaction of Aryl Alkyl Ketones with Bis(2,2,2-trifluoroethyl)phosphonoacetic Acid,
Tetrahedron Letters, Vol.44, No.49, 8853-8855, 2003.
(DOI: 10.1016/j.tetlet.2003.09.185,   CiNii: 1574231876485832704)
42. Shigeki Sano, Kenji Yokoyama, Motoo Shiro and Yoshimitsu Nagao :
A Facile Method for the Stereoselective Horner-Wadsworth-Emmons Reaction of Aryl Alkyl Ketones,
Chemical & Pharmaceutical Bulletin, Vol.50, No.5, 706-709, 2002.
(DOI: 10.1248/cpb.50.706,   CiNii: 1390282679140850688)
43. Yoshimitsu Nagao, Satoshi Miyamoto, Kazuhiko Hayashi, Ado Mihira and Shigeki Sano :
Synthesis of New Chiral Sulfinyldiacetic Acid Derivatives and Attempt at Chemoselective Asymmetric Pummerer Reaction,
Chemical & Pharmaceutical Bulletin, Vol.50, No.4, 558-562, 2002.
(DOI: 10.1248/cpb.50.558,   PubMed: 11964012,   CiNii: 1390282679140236032)
44. Yoshimitsu Nagao, Hitoshi Iimori, Satoru GOTO, Terukage Hirata, Shigeki Sano, Hiroshi Chuman and Motoo Shiro :
Remarkable Discrepancy in the Predominant Structures of Acyl(or Thioacyl)aminothiadiazoles, Acyl(or Thioazyl)aminooxadiazoles and Related Compounds Having the Potential for Rotational, Geometrical and Tautomeric Isomerism,
Tetrahedron Letters, Vol.43, No.9, 1709-1712, 2002.
(DOI: 10.1016/S0040-4039(02)00080-1,   Elsevier: Scopus)
45. Yoshimitsu Nagao, Akiharu Ueki, Kazunori Asano, Satoru Tanaka, Shigeki Sano and Motoo Shiro :
Facile Palladium(0)-Catalyzed Ring Expansion Reactions of Hydroxy Methoxyallenyl Cyclic Compounds via Hydropalladation,
Organic Letters, Vol.4, No.3, 455-457, 2002.
(DOI: 10.1021/ol010287k,   PubMed: 11820903)
46. Yoshimitsu Nagao, Satoshi Miyamoto, Kazuhiko Hayashi, Ado Mihira and Shigeki Sano :
Highly Chemoselective Pummerer Reactions of Sulfinyldiacetic Acid Derivative,
Tetrahedron Letters, Vol.43, No.8, 1519-1522, 2002.
(DOI: 10.1016/S0040-4039(02)00051-5)
47. Shigeki Sano, Kenji Yokoyama, Rie Teranishi, Motoo Shiro and Yoshimitsu Nagao :
Enantioselective Horner-Wadsworth-Emmons Reaction for the Asymmetric Synthesis of α-Fluoro-α,β-unsaturated Esters,
Tetrahedron Letters, Vol.43, No.2, 281-284, 2002.
(DOI: 10.1016/S0040-4039(01)02135-9,   Elsevier: Scopus)
48. Shigeki Sano, Tomoka Takehisa, Shiho Ogawa, Kenji Yokoyama and Yoshimitsu Nagao :
Stereoselective Synthesis of Tetrasubstituted (Z)-Alkenes form Aryl Alkyl Ketones Utilizing the Horner-Wadsworth-Emmons Reaction,
Chemical & Pharmaceutical Bulletin, Vol.50, No.9, 1300-1302, 2002.
49. Shigeki Sano, Rie Teranishi and Yoshimitsu Nagao :
Toward (Z)-Selective Horner-Wadsworth-Emmons Reaction of Aldehydes with 2-Fluoro-2-diethylphosphonoacetic Acid,
Tetrahedron Letters, Vol.43, No.50, 9183-9186, 2002.
(DOI: 10.1016/S0040-4039(02)02269-4,   CiNii: 1570572701769310080)
50. Yoshimitsu Nagao, Hitoshi Iimori, Hong Ki Nam, Shigeki Sano and Motoo Shiro :
Synthesis and Antibacterial Activity of New 1β-Methylcarbapenems Having the Potential for Intramolecular Nonbonded S---O Interactions,
Chemical & Pharmaceutical Bulletin, Vol.49, No.12, 1660-1661, 2001.
(DOI: 10.1248/cpb.49.1660,   PubMed: 11767095,   Elsevier: Scopus)
51. Norio Nakazawa, Keiko Tagami, Hitoshi Iimori, Shigeki Sano, Tsutomu Ishikawa and Yoshimitsu Nagao :
Copper(I) Iodine-Promoted Hydroxylation onto the Lithium or Potassium Enolate of Lactones and Lactams,
Heterocycles, Vol.55, No.11, 2157-2170, 2001.
(Elsevier: Scopus)
52. Shigeki Sano, Toshio Miwa, Kazuhiko Hayashi, Kazuo Nozaki, Yohei Ozaki and Yoshimitsu Nagao :
Chemoenzymatic Total Synthesis of (+)-Conagenin, a Low-molecular-weight Immunomodulator,
Tetrahedron Letters, Vol.42, No.24, 4029-4031, 2001.
(DOI: 10.1016/S0040-4039(01)00649-9,   CiNii: 1573950399809111680,   Elsevier: Scopus)
53. Keiko Tagami, Norio Nakazawa, Shigeki Sano and Yoshimitsu Nagao :
Asymmetric Syntheses of (+)-Camptothecin and (+)-7-Ethyl-10-methoxycamptothecin,
Heterocycles, Vol.53, No.4, 771-775, 2000.
(Elsevier: Scopus)
54. Yoshimitsu Nagao, Shigeki Sano, Kenji Morimoto, Hisao Kakegawa, Tadanobu Takatani, Motoo Shiro and Nobuhiko Katunuma :
Synthesis of a New Class of Cathepsin B Inhibitors Exploiting a Unique Reaction Cascade,
Tetrahedron Letters, Vol.41, No.14, 2419-2424, 2000.
55. Yoshimitsu Nagao, Hiroaki Nishijima, Hitoshi Iimori, Hideki Ushirogochi, Shigeki Sano and Motoo Shiro :
Desulfurilative Self-Coupling Reaction of 1,3-Thiazolidine-2-thiones and Intramolecular Non-Bonded S---S Interaction in the Crystallographic Structure of the Products,
Journal of Organometallic Chemistry, Vol.611, No.1/2, 172-177, 2000.
56. Shigeki Sano, Takahiro Ishii, Toshio Miwa and Yoshimitsu Nagao :
Tin-Mediated Enantioselective Aldol-Type Reaction for the Asymmetric Synthesis of α-Substituted Serines Utilizing an External Chiral Ligand, (-)-Sparteine,
Tetrahedron Letters, Vol.40, No.15, 3013-3016, 1999.
57. Ill-Yun Jeong, Woo-Song Lee, Satoru GOTO, Shigeki Sano, Motoo Shiro and Yoshimitsu Nagao :
Novel hetrocyclic ring-expansion and/or dehydration-hydration reactions of propargylic and allenylic hydroxy γ-lactams in the presence of strong base or Lewis acid,
Tetrahedron, Vol.54, No.48, 14437-14454, 1998.
58. Shigeki Sano, Tsuyoshi Ando, Kenji Yokoyama and Yoshimitsu Nagao :
New Reaction Mode of the Horner-Wadsworth-Emmons Reaction for the Preparation of α-Fluoro-α,β-unsaturated Esters,
Synlett, Vol.1998, No.7, 777-779, 1998.
(DOI: 10.1055/s-1998-1780)
59. Yoshimitsu Nagao, Terukage Hirata, Satoru GOTO, Shigeki Sano, Akikazu Kakehi, Kinji Iizuka and Motoo Shiro :
Intramolecular Nonbonded S---O Interaction Recognized in (Acylimino)thiadiazoline Derivatives as Angiotensin II Receptor Antagonists and Related Compounds,
Journal of the American Chemical Society, Vol.120, No.13, 3104-3110, 1998.
60. Yoshimitsu Nagao, Satoshi Tamai, Noriko Tanigawa, Shigeki Sano, Toshio Kumagai and Ikuo Kishi :
Synthesis and Antibacterial Activity of New, Non-natural 1β-Methylcarbapenem Bearing a σ-Symmetric Bicyclopyrazoliumthio Group as the Pendant Moiety,
Heterocycles, Vol.48, No.4, 617-620, 1998.
61. Shigeki Sano, Kazuhiko Hayashi, Toshio Miwa, Takahiro Ishii, Michiho Fujii, Hiromi Mima and Yoshimitsu Nagao :
New Enantiodivergent Procedure for the Syntheses of Chiral α-Substituted Serines from α-Alkyl-α-aminomalonates Utilizing Enzymatic Hydrolysis,
Tetrahedron Letters, Vol.39, No.31, 5571-5574, 1998.
62. Terukage Hirata, Hiromi Kogiso, Kenji Morimoto, Satoshi Miyamoto, Hiromi Taue, Shigeki Sano, Naoki Muguruma, Susumu Ito and Yoshimitsu Nagao :
Synthesis and Reactivities of 3-Indocyanine-green-acyl-1,3-thiazolidine-2-thione (ICG-ATT) as a New Near-Infrared Fluorescent-labeling Reagent,
Bioorganic & Medicinal Chemistry, Vol.6, No.11, 2179-2184, 1998.
63. Shigeki Sano, Maki Takebayashi, Toshio Miwa, Takahiro Ishii and Yoshimitsu Nagao :
Tin- or Magnesium-Mediated Diastereoselective Aldol-Type Reactions for the Asymmetric Synthesis of α-Substituted Serines,
Tetrahedron: Asymmetry, Vol.9, No.20, 3611-3614, 1998.
64. Shigeki Sano, Toshio Miwa, Xiao-Kai Liu, Takahiro Ishii, Tomoka Takehisa, Motoo Shiro and Yoshimitsu Nagao :
Tin- or Magnesium-Mediated Diastereoselective Aldol-Type Reactions for the Asymmetric Synthesis of α-Substituted Serines,
Tetrahedron: Asymmetry, Vol.9, No.20, 3615-3618, 1998.
65. Terukage Hirata, Satoru GOTO, Koichi Tamura, Masayasu Okuhira and Yoshimitsu Nagao :
Quantitative structure-activity relationships of benzoyliminothiadiazoline derivatives as angiotensin II receptor antagonists,
Bioorganic & Medicinal Chemistry Letters, Vol.7, No.4, 385-388, 1997.
66. Song Woo Lee, Ill-Yun Jeong, Motoo Shiro, Shigeki Sano and Yoshimitsu Nagao :
Efficient, Direct Synthesis of Novel Racemic Trimethoxy-Substituted [6] and,
Tetrahedron Letters, Vol.38, No.4, 611-614, 1997.
67. Shigeki Sano, Kenji Yokoyama, Mari Fukushima, Tetsuo Yagi and Yoshimitsu Nagao :
New Reaction Mode of the Horner-Wadsworth-Emmons Reaction Using Sn(OSO2CF3)2,
Chemical Communications, No.6, 559-560, 1997.
68. Keiko Tagami, Shuzo Takagi, Shigeki Sano, Motoo Shiro and Yoshimitsu Nagao :
Asymmetric Dihydroxylation onto the α,β-Unsaturated Carboxylic Ester Derivatives of Camptothecin,
Heterocycles, Vol.45, No.9, 1663-1669, 1997.
69. Kazuhiko Hayashi, Hiromi Kogiso, Shigeki Sano and Yoshimitsu Nagao :
Variable Stereoselectivity in the Imine Aldol Reactions Employing MgBr2 and Et3N,
Synlett, No.12, 1203-1205, 1996.
(DOI: 10.1055/s-1996-5721)
70. Masayuki Shibuya, Masakazu Wakayama, Yoshimitsu Naoe, Tadaaki Kawakami, Katsuya Ishigaki, Hisao Nemoto, Hisasi Shimizu and Yoshimitsu Nagao :
Cycloaromatization of enediyne model compounds via a reaction cascade triggered by hydrolysis of the a-alkynylmalonates,
Tetrahedron Letters, Vol.37, 865-868, 1996.
71. Yoshimitsu Nagao, Ill-Yun Jeong, Song Woo Lee and Shigeki Sano :
A New Ring Enlargement Reaction of γ-Lactones to Seven-Membered Cyclic Ethers via,
Chemical Communications, No.1, 19-20, 1996.
72. Yoshimitsu Nagao, Kweon Kim, Shigeki Sano, Hisao Kakegawa, Song Woo Lee, Hisashi Shimizu, Motoo Shiro and Nobuhiko Katunuma :
Syntheses and Reactions of the Diethyl α-Alkynylmalonates Involving the Generation of,
Tetrahedron Letters, Vol.37, No.6, 861-864, 1996.
73. Shigeki Sano, Hideki Ushirogochi, Kenji Morimoto, Satoshi Tamai and Yoshimitsu Nagao :
A New Enantiodivergent Procedure Utilising the Chemoselective Dieckmann-Type,
Chemical Communications, No.15, 1775-1776, 1996.
74. Masaru Kihara, Ikeuchi Motoki and Yoshimitsu Nagao :
Synthesis and Biological Evaluation of 3,4-Diphenyl-1,2-dihydroisoquinolines as a New Tamoxifen Analogue,
Drug Design and Discovery, Vol.12, No.3, 259-271, 1995.
(PubMed: 7662832)
75. Masaru Kihara, Ikeuchi Motoki, Yoshimitsu Nagao, Moritoki Hideki and Taira Zenei :
Synthesis and Enantioselectivity of Optically Active 1- and 3-Substituted 4-Phenyl-1,2,3,4-tetrahydroisoquinolin-4-ols and Related Compounds as Norepinephrine Potentiators,
Chemical & Pharmaceutical Bulletin, Vol.43, No.9, 1543-1546, 1995.
76. Masaru Kihara, Iwai Yasumasa and Yoshimitsu Nagao :
A New Synthesis of 3-Substituted Indolines and Indoles,
Heterocycles, Vol.41, No.10, 2279-2287, 1995.
77. Satoshi Tamai, Hideki Ushirogochi, Shigeki Sano, Yoshimitsu Nagao and Yoshimitsu Nagao :
New Reaction Mode of the Dieckmann-Type Cyclization under the Lewis Acid-Et3N,
Chemistry Letters, No.4, 295-296, 1995.
78. Shigeki Sano, Yoshimaro Kobayashi, Tatsuya Kondo, Maki Takebayashi, Shigeki Maruyama, Tetsuro Fujita and Yoshimitsu Nagao :
Asymmetric Total Synthesis of ISP-I (Myriocin, Thermozymocidin), a Potent,
Tetrahedron Letters, Vol.36, No.12, 2097-2100, 1995.
79. Shigeki Sano, Xiao-Kai Liu, Maki Takebayashi, Yoshimaro Kobayashi, Keiko Tabata, Motoo Shiro and Yoshimitsu Nagao :
Lewis Acid- and Cationic Lithium-Mediated Diastereoselective Aldol-Type Reaction Based,
Tetrahedron Letters, Vol.36, No.23, 4101-4104, 1995.
80. Masaru Kihara, Kashimoto Minoru, Kobayashi Yoshimaro, Yoshimitsu Nagao and Moritoki Hideki :
New Norepinephrine Potentiators:Synthesis and Structure-Activity Relationships of a series of 4-Phenyl-1,2,3,4-tetrahydroisoquinolin-4-ols,
Chemical & Pharmaceutical Bulletin, Vol.42, No.1, 67-73, 1994.
81. Masaru Kihara, Ikeuchi Motoki, Kobayashi Yoshimaro, Yoshimitsu Nagao and Moritoki Hideki :
Synthesis and Pharmacological Evaluation of Phenolic 2-Methyl-4-phenyl-1,2,3,4-tetrahydroisoquinolin-4-ols,
Drug Design and Discovery, Vol.11, 175-183, 1994.
82. Masaru Kihara, Xu Lai, Konishi Keiji, Yoshimitsu Nagao and Kobayashi Shigeru :
Isolation and Structure Elucidation of a Novel Alkaloid, Incartine, a Supposed Biosynthetic Intermediate, from Flowers of Lycoris incarnata,
Chemical & Pharmaceutical Bulletin, Vol.42, No.2, 289-292, 1994.
83. Yoshimitsu Nagao, Song Woo Lee, Yoichi Komaki, Shigeki Sano and Motoo Shiro :
New Six- to Eight-Membered-Ring Formation Based on the Intramolecular Endo- Mode,
Chemistry Letters, No.3, 597-600, 1994.
84. Satoshi Tamai, Satoru Miyauchi, Chikako Morizane, Kaname Miyagi, Hisashi Shimizu, Masaharu Kume, Shigeki Sano, Motoo Shiro and Yoshimitsu Nagao :
Enzymatic Hydrolyses of the σ-Symmetric Dicarboxylic Diesters Bearing a Sulfinyl Group,
Chemistry Letters, No.12, 2381-2384, 1994.
85. Shigeki Sano, Michiko Tanba and Yoshimitsu Nagao :
A Facile Synthesis of New Prostaglandin Analogues by Utilizing the Characteristics of the,
Heterocycles, Vol.38, No.3, 481-486, 1994.
86. Yoshimitsu Nagao, Kweon Kim, Yoichi Komaki, Shigeki Sano, Masaru Kihara and Motoo Shiro :
One-Pot Synthesis of New 1,3-Imidazolidines Possessing Three Aryl Groups via a 1,3-,
Heterocycles, Vol.38, No.3, 587-593, 1994.
87. Yoshimitsu Nagao, Shigeki Sano, Satoshi Nakagawa, Masanobu Suzuki, Motoo Shiro, Masaru Kido and Takao Nishi :
Synthesis of New Molecules Adopting a Unique Sigmoid Conformation with Stacked,
Heterocycles, Vol.36, No.8, 1715-1720, 1993.
88. Yoshimitsu Nagao, Shigeki Sano, Satoshi Nakagawa, Miho Tanaka, Motoo Shiro and Tohru Taga :
Characterization of the Sulfonic Esters Adopting a Folded Conformation with Stacked,
Chemistry Letters, No.6, 915-918, 1992.
89. Yoshimitsu Nagao, Jamal Mustafa, Shigeki Sano, Masahito Ochiai, Tazuko Tashiro and Shigeru Tsukagoshi :
Different Mechanisms of Action of Long Chain Fatty Acid Esters of Podophyllotoxin and,
Medicinal Chemistry Research, Vol.1, No.4, 295-299, 1991.
90. Yoshimitsu Nagao, Shigeki Sano, Masahito Ochiai and Eiichi Fujita :
Biomimetic, Chemical, and Spectroscopic Evaluations for the Radiosensitizing Potential of,
Tetrahedron, Vol.46, No.9, 3211-3232, 1990.
91. Yoshimitsu Nagao, Shigeki Sano, Masahito Ochiai, Kaoru Fuji, Sei-ichi Nishimoto, Tsutomu Kagiya, Chieko Murayama, Tomoyuki Mori, Yuta Shibamoto, Keisuke Sasai and Mitsuyuki Abe :
Radiosensitizing Hypoxic Cells with New 3-Nitro-1,2,4-triazole Derivatives in Vitro and,
Chemical & Pharmaceutical Bulletin, Vol.37, No.7, 1951-1953, 1989.
92. Chieko Murayama, Yoshimitsu Nagao, Shigeki Sano, Masahito Ochiai, Kaoru Fuji, Eiichi Fujita and Tomoyuki Mori :
Effect of Oridonin, a Rabdosia Diterpenoid, on Radiosensitization with Misonidazole,
Experientia, Vol.43, No.11/12, 1221-1223, 1987.

Academic Paper (Unrefereed Paper):

1. Yoshimitsu Nagao, Shigeki Sano, Masahito Ochiai, Kaoru Fuji, Sei-ichi Nishimoto, Tsutomu Kagiya, Yuta Shibamoto, Mitsuyuki Abe, Chieko Murayama and Tomoyuki Mori :
Synthetic Development of Hypoxic Cell Sensitizers Having 3-Nitrotriazole Moiety,
Journal of Pharmacobio-Dynamics, Vol.10, s-155, 1987.
2. Yoshimitsu Nagao, Shigeki Sano, Tadayo Miyasaka, Masahito Ochiai, Kaoru Fuji, Eiichi Fujita and Hisashi Ishii :
Evaluation of the Affinity of New N Atom-Containing Tumor Inhibitors for Nucleic Acids,
Nucleic Acids Research, Symposium Series, Vol.16, 37-40, 1985.

Review, Commentary:

1. Susumu Ito, Naoki Muguruma, Tetsuo Kimura, Hiromi Yano, Yoshitaka Imoto, Koichi Okamoto, Masako Kaji, Shigeki Sano and Yoshimitsu Nagao :
Principle and Clinical Usefulness of the Infrared Fluorescence Endoscopy,
The Journal of Medical Investigation : JMI, Vol.53, No.1/2, 1-8, Feb. 2006.
(Tokushima University Institutional Repository: 110782,   DOI: 10.2152/jmi.53.1,   PubMed: 16537990)
2. Yoshimitsu Nagao and Shigeki Sano :
Cyclization, Ring Expansion, and Several Cascade Reactions Utilizing Allenylic Molecular Structure Characteristics,
Journal of Synthetic Organic Chemistry, Japan, Vol.61, No.11, 1088-1098, Nov. 2003.
(DOI: 10.5059/yukigoseikyokaishi.61.1088,   CiNii: 1390282680287473024,   Elsevier: Scopus)
3. Susumu Ito, Naoki Muguruma, 林 重仁, 日下 至弘, 多田津 昌也, 多田津 陽子, Koichi Okamoto, 井本 佳孝, 稲山 久美, 板東 輝実, 田岡 聡子, 高川 真由子, 矢野 充保, 伊井 邦雄, Yoshimitsu Nagao, Shigeki Sano, 芝村 誠一, 島田 典招, 石田 和彦 and 中村 一成 :
赤外線蛍光内視鏡の原理と応用,
Biomedical THERMOLOGY, Vol.23, 77-97, 2003.
4. Shigeki Sano and Yoshimitsu Nagao :
Asymmetric Synthesis of a-Substituted Serines,
Journal of Synthetic Organic Chemistry, Japan, Vol.58, No.8, 756-765, 2000.

Proceeding of International Conference:

1. Chung Keun Jin, Toshiaki Yamada, Takashi Masuda, Yoshimitsu Nagao and Shigeki Sano :
Synthesis of rac-Alkynylfluorosilanes and Their Application Reactions,
Post ISOS XV Symposium, Takasaki, Jun. 2008.
2. Michiyasu Nakao, Masanori Takeyasu, Shigeki Sano and Yoshimitsu Nagao :
Synthesis of Optical Active Diketopiperazines for Absolute Configuration Determination of α-Amino Acids,
The 12th Japan-Korea Joint Symposium on Drug Design and Development, Sendai, May 2008.
3. Chung Keun Jin, Toshiaki Yamada, Shigeki Sano and Yoshimitsu Nagao :
Synthesis of Dialkynyldiarylsilanes and Their Application Reactions,
The Winter School of Sokendai/Asian CORE Program Frontiers of Materials, Photo-, and Theoretical Molecular Sciences, Okazaki, Jan. 2008.
4. Shigeki Sano, Etsuko Harada and Yoshimitsu Nagao :
Novel Synthesis of β,γ-Unsaturated Esters Utilizing Tandem Double Bond Migration-Esterification,
Seoul National University-The University of Tokushima Young Medicinal Chemist Symposium - Recent Status and Future Prospect of Medicinal Chemistry, Seoul, Jul. 2005.
5. Shigeki Sano, Eiko Kujime and Yoshimitsu Nagao :
Synthesis of Chiral Phosphonoacetates as Novel Horner-Wadsworth-Emmons Reagents,
Seoul National University-The University of Tokushima Young Medicinal Chemist Symposium - Recent Status and Future Prospect of Medicinal Chemistry, Seoul, Jul. 2005.
6. Shigeki Sano, Shinobu Abe and Yoshimitsu Nagao :
Asymmetric Horner-Wadsworth-Emmons Reaction Utilizing Isomannide Derivatives as Chiral Auxiliaries,
Seoul National University-The University of Tokushima Young Medicinal Chemist Symposium - Recent Status and Future Prospect of Medicinal Chemistry, Seoul, Jul. 2005.
7. Kazuhiko Hayashi, Yoshifumi Ikee, Shigeki Sano and Yoshimitsu Nagao :
Synthesis of the Pendant Moiety of Oral 1β-Methylcarbapenem Antibiotic L-084 Using 1-Azabicyclo[1.1.0]butane,
Seoul National University-The University of Tokushima Young Medicinal Chemist Symposium - Recent Status and Future Prospect of Medicinal Chemistry, Seoul, Jul. 2005.
8. Motoyuki Miyamoto, Shigeki Sano and Yoshimitsu Nagao :
Investigation of Stereoselective Asymmetric Pummerer Reaction and Pummerer-type Cyclization,
Seoul National University-The University of Tokushima Young Medicinal Chemist Symposium - Recent Status and Future Prospect of Medicinal Chemistry, Seoul, Jul. 2005.
9. Noriaki Tanimoto, Takashi Honjo, Shigeki Sano and Yoshimitsu Nagao :
Catalytic Enantioselective Thiolysis of Prochiral Cyclic Dicarboxylic Anhydrides Utilizing Cinchona Alkaloids,
Seoul National University-The University of Tokushima Young Medicinal Chemist Symposium - Recent Status and Future Prospect of Medicinal Chemistry, Seoul, Jul. 2005.
10. Takashi Honjo, Shigeki Sano and Yoshimitsu Nagao :
Highly Enantioselective Catalytic Thiolysis of Prochiral Cyclic Dicarboxylic Anhydrides,
Seoul National University-The University of Tokushima Young Medicinal Chemist Symposium - Recent Status and Future Prospect of Medicinal Chemistry, Seoul, Jul. 2005.
11. Jin Keun Chung, Shigeki Sano and Yoshimitsu Nagao :
Development of an Improved Synthetic Method for Monosubstituted Alkynylfluorosilanes,
Seoul National University-The University of Tokushima Young Medicinal Chemist Symposium - Recent Status and Future Prospect of Medicinal Chemistry, Seoul, Jul. 2005.
12. Shigeki Sano, Michiyasu Nakao and Yoshimitsu Nagao :
Novel Enantiodivergent Synthesis of α-Methylserine Derivatives Utilizing Enzymatic Acetylation,
Seoul National University-The University of Tokushima Young Medicinal Chemist Symposium - Recent Status and Future Prospect of Medicinal Chemistry, Seoul, Jul. 2005.
13. Shigeki Sano, Yoko Kuroda and Yoshimitsu Nagao :
Toward Synthesis of Dipeptide-Mimetics Based on Fluoroolefin Isosteres,
Seoul National University-The University of Tokushima Young Medicinal Chemist Symposium - Recent Status and Future Prospect of Medicinal Chemistry, Seoul, Jul. 2005.
14. Shigeki Sano and Yoshimitsu Nagao :
New Aspects of the Horner-Wadsworth-Emmons Reaction of Phosphonoacetic Acids,
14th International Symposium on Fine Chemistry and Functional Polymers, Hohhot, Inner Mongolia, China, Aug. 2004.
15. Kazuhiko Hayashi, Yoshifumi Ikee, Shigeki Sano and Yoshimitsu Nagao :
Synthesis of the Pendant Moiety of Oral 1β-Methylcarbapenem Antibiotic L-084 Using 1-Azabicyclo[1.1.0]butane,
Pharmaceutical Sciences World Congress, Kyoto, May 2004.
16. Motoyuki Miyamoto, Shigeki Sano and Yoshimitsu Nagao :
Investigation of Stereoselective Asymmetric Pummerer Reaction and Pummerer-Type Cyclization,
Pharmaceutical Sciences World Congress, Kyoto, May 2004.
17. Takashi Honjo, Shigeki Sano and Yoshimitsu Nagao :
Syntheses and Characterization of Thiazole Derivatives Having the Potential for Intramolecular Nonbonded Interactions,
Pharmaceutical Sciences World Congress, Kyoto, May 2004.
18. Satoru Tanaka, Masunori Kumazawa, Shigeki Sano and Yoshimitsu Nagao :
Development of Ring-Expansion Reactions Using Hydroxy Methoxyallenyl or Propenoyl Cyclic Compounds,
Pharmaceutical Sciences World Congress, Kyoto, May 2004.
19. Shigeki Sano and Yoshimitsu Nagao :
Stereoselective Synthesis of (Z)-fluoroolefins: (s-Z)-Amide isosteres,
Pharmaceutical Sciences World Congress, Kyoto, May 2004.
20. Kazuhiko Hayashi, Yoshifumi Ikee, Shigeki Sano and Yoshimitsu Nagao :
Synthesis of the Pendant Moiety of Oral 1b-Methylcarbapenem Antibiotics L-084,
The 10th Korea-Japan Joint Symposium on Drug Design and Development, Tokushima, Apr. 2004.
21. Shigeki Sano and Yoshimitsu Nagao :
Synthesis of P-Chiral Phosphonates: Novel Horner-Wadsworth-Emmons Reagents,
The 10th Korea-Japan Joint Symposium on Drug Design and Development, Tokushima, Apr. 2004.
22. Shigeki Sano and Yoshimitsu Nagao :
HWE Reaction of Phosphonoacetic Acids and Synthesis of Novel P-Chiral HWE Reagents,
The 2nd Takeda Science Foundation Symposium on PharmaSciences, Kyoto, Dec. 2003.
23. Shigeki Sano and Yoshimitsu Nagao :
Stereoselective Horner-Wadsworth-Emmons Reaction for the Synthesis of Amide Isosteres,
Fifth AFMC International Medicinal Chemistry Symposium, Kyoto, Japan, Oct. 2003.
24. Shigeki Sano and Yoshimitsu Nagao :
Tandem Reduction-Olefination for the Stereoselective Synthesis of (Z)-α-Fluoro-α,β-unsaturated Esters,
The 9th Korea-Japan Joint Symposium on Drug Design and Development, Seoul, May 2002.
25. Yoshimitsu Nagao, Akiharu Ueki, Kazunori Asano, Satoru Tanaka and Shigeki Sano :
Palladium(0)-Catalyzed Ring-Expansion Reactions of Allenyl Alcohol Derivatives,
The Joint Symposium between Seoul National University and University of Tokushima on Pharmacy, Cheju Island, Aug. 2000.
26. Yoshimitsu Nagao and Shigeki Sano :
Characterization of the Organosulfur Compound Bearing S---X (X = O, N, Br, and p) Close Contact and Its Application to Organic Reactions,
4th Australia-Japan Joint Symposium on Drug Design and Development, Melbourne, May 2000.
27. Yoshimitsu Nagao and Shigeki Sano :
Characterization of the Organosulfur Compound Bearing S---X (X = O, N, Br, and p) Close Contact and Its Application to Organic Reactions,
4th Australia-Japan Joint Symposium on Drug Design and Development, Melbourne, May 2000.
28. Shigeki Sano and Yoshimitsu Nagao :
Asymmetric Total Synthesis of (+)-Conagenin,
4th Australia-Japan Joint Symposium on Drug Design and Development, Melbourne, May 2000.
29. Shigeki Sano, Tomoka Takehisa and Yoshimitsu Nagao :
Stereoselective Synthesis of Ozagrel Derivatives Utilizing HWE Reaction,
The 7th Korea-Japan Joint Symposium on Drug Design and Development, Busan, May 1999.
30. Yoshimitsu Nagao, Hiroe Takeshige, Ado Mihira and Shigeki Sano :
Optical Resolution of Racemic S-Oxothiodiglycolic Acid by Exploiting a Chiral Thiazolidine-2-thione,
The 7th Korea-Japan Joint Symposium on Drug Design and Development, Busan, May 1999.
31. Yoshimitsu Nagao, Satoshi Miyamoto and Shigeki Sano :
Chemo- and Enantioselective Pummerer-type Reaction of Chiral Sulfoxides Having Potential S---O Interactions,
The 7th Korea-Japan Joint Symposium on Drug Design and Development, Busan, May 1999.
32. Yoshimitsu Nagao, Hitoshi Iimori, Satoru GOTO and Shigeki Sano :
Synthesis of New Organosulfur Compounds Having Potential for Intra- or Intermolecular Nonbonded S---X (O, N, S, etc.) Interactions,
The 7th Korea-Japan Joint Symposium on Drug Design and Development, Busan, May 1999.
33. Shigeki Sano, Toshio Miwa and Yoshimitsu Nagao :
Asymmetric Total Synthesis of (+)-Conagenin,
The 7th Korea-Japan Joint Symposium on Drug Design and Development, Busan, May 1999.
34. Yoshimitsu Nagao, Kenji Morimoto and Shigeki Sano :
Synthesis of New Cysteine Protease Inhibitors Bearing L-Valine,
The 7th Korea-Japan Joint Symposium on Drug Design and Development, Busan, May 1999.
35. Yoshimitsu Nagao, Norio Nakazawa and Shigeki Sano :
Development of Hydroxylation at the α-Position of Carbonyl Compounds,
The 7th Korea-Japan Joint Symposium on Drug Design and Development, Busan, May 1999.
36. Shigeki Sano and Yoshimitsu Nagao :
New Approach to the Stereoselective Horner-Wadsworth-Emmons Reaction,
The 7th Korea-Japan Joint Symposium on Drug Design and Development, Busan, May 1999.
37. Shigeki Sano, Takahiro Ishii and Yoshimitsu Nagao :
Highly Enantioselective Synthesis of α-Substituted Serine Derivatives Utilizing a Chiral Ligand,
3rd Australia-Japan Symposium on Drug Design and Development, Naruto, Sep. 1998.
38. Shigeki Sano, Kenji Yokoyama and Yoshimitsu Nagao :
New Approach to the Stereoselective Horner-Wadsworth-Emmons Reaction,
3rd Australia-Japan Symposium on Drug Design and Development, Naruto, Sep. 1998.
39. Yoshimitsu Nagao, Satoru GOTO and Shigeki Sano :
Intramolecular Nonbonded S---X (X = O, N, S) Interaction Recognized in Several Drugs,
3rd Australia-Japan Symposium on Drug Design and Development, Naruto, Sep. 1998.
40. Yoshimitsu Nagao, Terukage Hirata, Satoru GOTO and Shigeki Sano :
Intramolecular nonbonded S---O interaction recognized in acyliminothiadiazoline derivatives as angiotensin II receptor antagonists and other drugs,
The 6th Korea/Japan Symposium on Drug Design and Development, Tokyo, Jan. 1998.
41. Shigeki Sano and Yoshimitsu Nagao :
Asymmetric Synthesis of α-Substituted Serine Derivatives,
The 5th China-Japan Joint Symposium on Drug Design and Development, Chengdu, Sep. 1997.
42. Yoshimitsu Nagao, Terukage Hirata, Satoru GOTO, Shigeki Sano and Motoo Shiro :
Aspects for 1,5-type S---O nonbonded interaction observed in acyliminothiadiazoline derivatives as angiotensin II receptor antagonists,
AIMECS 97 AFMC International Medicinal Chemistry Symposium, Seoul, Jan. 1997.
43. Shigeki Sano and Yoshimitsu Nagao :
Design and Synthesis of New Cysteine Protease Inhibitors,
The 2nd Australia-Japan Joint Symposium on Drug Design and Developmant, Cairns, Sep. 1996.
44. Terukage Hirata, J. Nomiyama, N. Sakae, K. Nishimura, M. Yokomoto, S. Inoue, K. Tamura, M. Okuhira, H. Amano, Satoru GOTO and Yoshimitsu Nagao :
New angiotensin II receptor antagonists: Syntheses and biological properties, and structure-activity relationships,
The 2nd Australia/Japan Symposium on Drug Design and Development, North Queensland, Jan. 1996.

Proceeding of Domestic Conference:

1. Michiyasu Nakao, Masanori Takeyasu, Yuriko Toriuchi, Yoshimitsu Nagao and Shigeki Sano :
N-Methyldiketopiperazine Catalyzed Direct Asymmetric Aldol Reaction,
日本薬学会第132年会, Mar. 2012.
2. Masanori Kamura, Takeshi Tsumura, Michiyasu Nakao, Shigeki Sano and Yoshimitsu Nagao :
環状酸無水物の不斉アルコリシスを基盤とする光学活性フタラジノンの合成,
第48回日本薬学会・日本薬剤師会・日本病院薬剤師会中国四国支部学術大会, Nov. 2009.
3. Takashi Ichikawa, Michiyasu Nakao, Shigeki Sano and Yoshimitsu Nagao :
DCCを用いるα,β-不飽和カルボン酸の脱共役エステル化反応,
第48回日本薬学会・日本薬剤師会・日本病院薬剤師会中国四国支部学術大会, Nov. 2009.
4. Takeshi Tumura, Masashi Horibe, Michiyasu Nakao, Shigeki Sano and Yoshimitsu Nagao :
σ対称環状炭酸エステルの触媒的エナンチオ選択的開環反応,
第48回日本薬学会・日本薬剤師会・日本病院薬剤師会中国四国支部学術大会, Nov. 2009.
5. Michiyasu Nakao, Yuta Hiroyama, Shigeki Sano and Yoshimitsu Nagao :
芳香環含有ジケトピペラジン類のコンホメーション解析,
第48回日本薬学会・日本薬剤師会・日本病院薬剤師会中国四国支部学術大会, Nov. 2009.
6. Takashi Ichikawa, Michiyasu Nakao, Shigeki Sano and Yoshimitsu Nagao :
Deconjugative Esterification of α,β-Unsaturated Carboxylic Acids through Carbodiimide Coupling,
第35回反応と合成の進歩シンポジウム, Nov. 2009.
7. Akinobu Morimoto, Shigeki Sano, Yoshimitsu Nagao and Hiro-O Ito :
Synthetic Development of Methanethiol-Trapping Agents,
日本薬学会第129年会, Mar. 2009.
8. Hiroshi Nanataki, Shigeki Sano and Yoshimitsu Nagao :
Synthesis of AA-Ψ[(Z)-CF=C]-Pro via Horner-Wadsworth-Emmons Reaction,
日本薬学会第129年会, Mar. 2009.
9. Takashi Ichikawa, Michiyasu Nakao, Shigeki Sano and Yoshimitsu Nagao :
Deconjugative Esterification of 2-Cyclohexylideneacetic Acids with Intramolecular Chiral Transfer,
日本薬学会第129年会, Mar. 2009.
10. Takeshi Tsumura, Shigeki Sano and Yoshimitsu Nagao :
Catalytic Asymmetric Desymmetrization of σ-Symmetric 1,3-Diols,
日本薬学会第129年会, Mar. 2009.
11. Michiyasu Nakao, Masanori Takeyasu, Yuta Hiroyama, Shigeki Sano and Yoshimitsu Nagao :
Synthesis of Diketopiperazines for Determining Absolute Configuration of α-Amino Acids (3),
日本薬学会第129年会, Mar. 2009.
12. Takeshi Tsumura, Shigeki Sano and Yoshimitsu Nagao :
シンコナアルカロイド誘導体を用いたσ対称1,3-ジオールの非対称化反応,
創薬懇話会2008, Dec. 2008.
13. Michiyasu Nakao, Masanori Takeyasu, Yuta Hiroyama, Shigeki Sano and Yoshimitsu Nagao :
複素環化合物の特性を活用したα-アミノ酸の簡便絶対配置決定法,
創薬懇話会2008, Dec. 2008.
14. Michiyasu Nakao, Masanori Takeyasu, Yuta Hiroyama, Shigeki Sano and Yoshimitsu Nagao :
Synthesis of Optical Active Diketopiperazines for Absolute Configuration Determination of α-Amino Acids,
第38回複素環化学討論会, Nov. 2008.
15. Akinobu Morimoto, Shigeki Sano, Yoshimitsu Nagao and Hiro-O Ito :
揮発性チオール捕捉反応剤の合成開発研究,
第47回日本薬学会·日本薬剤師会·日本病院薬剤師会中国四国支部学術大会, Nov. 2008.
16. Hiroshi Nanataki, Shigeki Sano and Yoshimitsu Nagao :
フルオロオレフィン型プロリン含有ジペプチドミメティクスの合成,
第47回日本薬学会·日本薬剤師会·日本病院薬剤師会中国四国支部学術大会, Nov. 2008.
17. Mai Kamino, Yukari Nakayama, Shigeki Sano and Yoshimitsu Nagao :
アンギバクチンならびにアンヒドロアンギバクチンの合成研究,
第47回日本薬学会·日本薬剤師会·日本病院薬剤師会中国四国支部学術大会, Nov. 2008.
18. Yukiko Ose, Shigeki Sano and Yoshimitsu Nagao :
ケトンの不斉還元によるフルオロオレフィン型光学活性ジペプチドミメティクスの合成,
第47回日本薬学会·日本薬剤師会·日本病院薬剤師会中国四国支部学術大会, Nov. 2008.
19. Takashi Ichikawa, Michiyasu Nakao, Shigeki Sano and Yoshimitsu Nagao :
カルボジイミド型脱水縮合剤を用いるケテン経由の脱共役エステル化反応,
第47回日本薬学会·日本薬剤師会·日本病院薬剤師会中国四国支部学術大会, Nov. 2008.
20. Takeshi Tsumura, Shigeki Sano and Yoshimitsu Nagao :
キラルスルホンアミド-亜鉛錯体を用いたσ対称1,3-ジオールの触媒的エナンチオ選択的アセチル化反応,
第47回日本薬学会·日本薬剤師会·日本病院薬剤師会中国四国支部学術大会, Nov. 2008.
21. Michiyasu Nakao, Masanori Takeyasu, Yuta Hiroyama, Shigeki Sano and Yoshimitsu Nagao :
1H NMRを用いるα-アミノ酸の簡便絶対配置決定法の開発,
第47回日本薬学会·日本薬剤師会·日本病院薬剤師会中国四国支部学術大会, Nov. 2008.
22. Takeshi Tsumura, Shigeki Sano and Yoshimitsu Nagao :
σ対称1,3-ジオールを基質とする触媒的エナンチオ選択的アセチル化反応,
第34回反応と合成の進歩シンポジウム, Nov. 2008.
23. Takeshi Tsumura, Shigeki Sano and Yoshimitsu Nagao :
キラルスルホンアミド-亜鉛錯体を用いるσ対称1,3-ジオールの不斉モノアシル化反応,
第24回若手化学者のための化学道場, Sep. 2008.
24. Mai Kamino, Yoshifumi Ikee, Kana Hashimoto, Shigeki Sano and Yoshimitsu Nagao :
Total Synthesis of Anguibactin,
日本薬学会第128年会, Mar. 2008.
25. Takashi Ichikawa, Michiyasu Nakao, Shigeki Sano and Yoshimitsu Nagao :
Deconjugative Esterification through Carbodiimide Coupling,
日本薬学会第128年会, Mar. 2008.
26. Michiyasu Nakao, Masanori Takeyasu, Saori Nakano, Shigeki Sano and Yoshimitsu Nagao :
Synthesis of Diketopiperazines for Absolute Configuration Determination of α-Amino Acids (2),
日本薬学会第128年会, Mar. 2008.
27. Michiyasu Nakao, 竹安 正範, 中野 沙織, Shigeki Sano and Yoshimitsu Nagao :
1H NMRを活用するα-アミノ酸誘導体の新規絶対配置決定法の開発,
第46回日本薬学会·日本薬剤師会·日本病院薬剤師会中国四国支部学術大会, Nov. 2007.
28. 山下 大輔, Shigeki Sano and Yoshimitsu Nagao :
2-アシル-2-ホスホノ酢酸エステルの合成とタンデム型還元-オレフィン化反応,
第46回日本薬学会·日本薬剤師会·日本病院薬剤師会中国四国支部学術大会, Nov. 2007.
29. Michiyasu Nakao, 竹安 正範, 中野 沙織, Shigeki Sano and Yoshimitsu Nagao :
光学活性ジケトピペラジンの合成とα-アミノ酸誘導体の新規絶対配置決定法の開発,
第33回反応と合成の進歩シンポジウム, Nov. 2007.
30. 井上 尚兵, 木下 陽子, 青柳 えり子, Naoki Muguruma, Susumu Ito, Shigeki Sano and Yoshimitsu Nagao :
新規ICG-ATT誘導体を用いた蛋白質標識モデル実験,
日本薬学会第127年会, Mar. 2007.
31. Yoko Kuroda, Yukiko Ose, Shigeki Sano and Yoshimitsu Nagao :
フルオロオレフィン型光学活性ジペプチドミメティクスの合成研究,
日本薬学会第127年会, Mar. 2007.
32. 陳 青根, Toshiaki Yamada, Motoyuki Miyamoto, Shigeki Sano and Yoshimitsu Nagao :
新規な1-シラアレン，シラシクロブテン，ならびに1,3-共役ジエンの合成,
日本薬学会第127年会, Mar. 2007.
33. Michiyasu Nakao, Masanori Takeyasu, Shigeki Sano and Yoshimitsu Nagao :
ジケトピペラジン構造を基盤とするα-アミノ酸の新規絶対配置決定法の開発研究,
日本薬学会第127年会, Mar. 2007.
34. Michiyasu Nakao, 竹安 正範, Shigeki Sano and Yoshimitsu Nagao :
α-置換セリン誘導体のエナンチオ分岐的合成と新規絶対配置決定法の開発,
第32回反応と合成の進歩シンポジウム, Dec. 2006.
35. 陳 青根, 山田 敏彰, Shigeki Sano and Yoshimitsu Nagao :
新規なジアリールジアルキニルシラン及びシラシクロブテンの合成ならびに応用研究,
第32回反応と合成の進歩シンポジウム, Dec. 2006.
36. 大久保 好規, Shigeki Sano, Yoshimitsu Nagao and 掛川 寿夫 :
HWE反応を用いるイソリクイリチゲニンならびにZ異性体の立体選択的合成,
第45回日本薬学会·日本病院薬剤師会中国四国支部学術大会, Oct. 2006.
37. 黒田 陽子, 大勢 祐希子, Shigeki Sano and Yoshimitsu Nagao :
ジペプチドイソステアCbz-AA1-Ψ[(Z)-CF=C]-AA2の合成研究,
第45回日本薬学会·日本病院薬剤師会中国四国支部学術大会, Oct. 2006.
38. Michiyasu Nakao, 竹安 正範, Shigeki Sano and Yoshimitsu Nagao :
α-置換セリン誘導体のエナンチオ分岐的化学-酵素合成ならびに絶対配置の決定,
第45回日本薬学会·日本病院薬剤師会中国四国支部学術大会, Oct. 2006.
39. Hirofumi Shibata, 近藤 京子, Kazuyoshi Kawazoe, Yoshihisa Takaishi, Yoshimitsu Nagao and Tomihiko Higuti :
MRSAに対するオクチルガレートの抗菌・抗アイルスマー活性に及ぼす金属イオンの影響,
第51回日本ブドウ球菌研究会, Sep. 2006.
40. 陳 青根, 山田 敏彰, Shigeki Sano and Yoshimitsu Nagao :
モノアルキニルシランとジアルキニルシランの合成開発及びその応用研究,
第7回長井長義記念シンポジウム, Sep. 2006.
41. 増田 隆司, 宮本 素行, Shigeki Sano and Yoshimitsu Nagao :
非結合性S•••O相互作用を基盤とする不斉Pummerer反応及び関連不斉識別反応への応用,
第7回長井長義記念シンポジウム, Sep. 2006.
42. 津村 武史, 本城 崇, Shigeki Sano and Yoshimitsu Nagao :
キラルスルホンアミドアミン触媒を用いたプロキラルな化合物の触媒的エナンチオ選択的非対称化反応の開発,
第7回長井長義記念シンポジウム, Sep. 2006.
43. 大久保 好規, Shigeki Sano, Yoshimitsu Nagao and 掛川 寿夫 :
イソリクイリチゲニンならびにZ異性体の効率的合成,
第7回長井長義記念シンポジウム, Sep. 2006.
44. 池江 克文, 橋本 佳奈, 上野 麻衣, 中島 正晃, 林 一彦, Shigeki Sano and Yoshimitsu Nagao :
アザビシクロブタンを活用するニューキノロン系抗菌剤の合成,
第7回長井長義記念シンポジウム, Sep. 2006.
45. 黒田 陽子, 大勢 祐希子, Shigeki Sano and Yoshimitsu Nagao :
ジペプチドイソステアCbz-Gly-Ψ[(Z)-CF=C]-Glyの立体選択的合成,
第7回長井長義記念シンポジウム, Sep. 2006.
46. 井上 尚兵, 木下 陽子, Shigeki Sano, Naoki Muguruma, Susumu Ito and Yoshimitsu Nagao :
新規な蛋白質標識試薬の合成開発研究,
第7回長井長義記念シンポジウム, Sep. 2006.
47. 久次米 永子, 田中 裕子, 林 一彦, 城 始勇, Shigeki Sano and Yoshimitsu Nagao :
不斉リン原子を有する新規ホスホノ酢酸エステルの化学-酵素合成,
第7回長井長義記念シンポジウム, Sep. 2006.
48. Michiyasu Nakao, 竹安 正範, 山本 千代, Shigeki Sano and Yoshimitsu Nagao :
α-置換セリン誘導体のエナンチオ分岐的化学-酵素合成,
第7回長井長義記念シンポジウム, Sep. 2006.
49. 陳 青根, 山田 敏彰, Shigeki Sano and Yoshimitsu Nagao :
異種ジアリールジアルキニル置換シラン及びシラシクロブテンの合成開発,
日本薬学会第126年会, Mar. 2006.
50. 宮本 素行, 増田 隆司, Shigeki Sano and Yoshimitsu Nagao :
非結合性S•••O相互作用を基盤とする不斉Pummerer反応及びアセチル化反応への応用,
日本薬学会第126年会, Mar. 2006.
51. 本城 崇, 津村 武史, Shigeki Sano and Yoshimitsu Nagao :
プロキラルな環状ジカルボン酸無水物の触媒的高エナンチオ選択的アルコリシス,
日本薬学会第126年会, Mar. 2006.
52. 井上 尚兵, Shigeki Sano and Yoshimitsu Nagao :
新規ICG-ATT標識化合物の合成開発,
日本薬学会第126年会, Mar. 2006.
53. 谷本 典昭, 本城 崇, Shigeki Sano and Yoshimitsu Nagao :
新規スルホンアミド触媒を用いたプロキラル環状ジカルボン酸無水物の不斉チオリシス及びアルコリシス,
日本薬学会第126年会, Mar. 2006.
54. 池江 克文, 橋本 佳奈, 中島 正晃, 林 一彦, Shigeki Sano and Yoshimitsu Nagao :
アザビシクロブタンを活用したニューキノロン系抗菌剤の合成,
日本薬学会第126年会, Mar. 2006.
55. Shigeki Sano, Michiyasu Nakao, 山本 千代 and Yoshimitsu Nagao :
リパーゼを用いるα-置換セリン誘導体のエナンチオ分岐的合成,
日本薬学会第126年会, Mar. 2006.
56. Shigeki Sano, 黒田 陽子 and Yoshimitsu Nagao :
Z型フルオロオレフィンを基盤とするジペプチドミメティクスの合成,
日本薬学会第126年会, Mar. 2006.
57. Shigeki Sano, 原田 悦子 and Yoshimitsu Nagao :
カルボジイミド系縮合試薬を用いるタンデム型二重結合転位-エステル化および-アミド化反応,
日本薬学会第126年会, Mar. 2006.
58. Shigeki Sano, 久次米 永子, 田中 裕子 and Yoshimitsu Nagao :
エステラーゼを用いる新規光学活性ホスホノ酢酸エステルの合成,
日本薬学会第126年会, Mar. 2006.
59. Yoshimitsu Nagao, 池江 克文, 橋本 佳奈, 中島 正晃, 林 一彦 and Shigeki Sano :
高歪み分子アザビシクロブタンを活用する抗菌剤合成,
第24回メディシナルケミストリーシンポジウム, Nov. 2005.
60. Shigeki Sano, 黒田 陽子 and Yoshimitsu Nagao :
Z選択的タンデム型還元-フルオロオレフィン化反応を用いるジペプチドミメティクスの合成,
第44回日本薬学会·日本病院薬剤師会中国四国支部学術大会, Nov. 2005.
61. Shigeki Sano, 原田 悦子 and Yoshimitsu Nagao :
2-シクロヘキシリデン酢酸類のタンデム型二重結合転位-エステル化反応,
第44回日本薬学会·日本病院薬剤師会中国四国支部学術大会, Nov. 2005.
62. Shigeki Sano, Michiyasu Nakao, 山本 千代 and Yoshimitsu Nagao :
酵素アシル化を用いるα-置換セリン誘導体のエナンチオ分岐的合成,
第44回日本薬学会·日本病院薬剤師会中国四国支部学術大会, Nov. 2005.
63. Shigeki Sano, 久次米 永子, 田中 裕子 and Yoshimitsu Nagao :
不斉リン原子を有する新規光学活性ホスホノ酢酸エステルの合成,
第44回日本薬学会·日本病院薬剤師会中国四国支部学術大会, Nov. 2005.
64. Shigeki Sano, 安部 忍 and Yoshimitsu Nagao :
軸性キラリティーを有する2-メチル-2-シクロヘキシリデン酢酸エステル類の合成,
第44回日本薬学会·日本病院薬剤師会中国四国支部学術大会, Nov. 2005.
65. 本城 崇, Shigeki Sano and Yoshimitsu Nagao :
新規キラルスルホンアミド触媒を用いたプロキラルなσ対称化合物の触媒的エナンチオ選択的非対称化,
第31回反応と合成の進歩シンポジウム, Nov. 2005.
66. 熊沢 益徳, 井上 尚兵, 田中 悟, Shigeki Sano and Yoshimitsu Nagao :
パラジウム触媒反応を活用するフラン環形成反応,
第6回長井長義記念シンポジウム, Jul. 2005.
67. 本城 崇, Shigeki Sano and Yoshimitsu Nagao :
新規なキラルスルホンアミド触媒を用いた環状ジカルボン酸無水物の触媒的高エナンチオ選択的チオリシス,
第6回長井長義記念シンポジウム, Jul. 2005.
68. Yoshimitsu Nagao, 熊沢 益徳, 井上 尚兵, 田中 悟 and Shigeki Sano :
パラジウム触媒反応を活用するフラン環形成反応,
日本薬学会第125年会, Mar. 2005.
69. Yoshimitsu Nagao, 池江 克文, 橋本 佳奈, 中島 正晃, 林 一彦 and Shigeki Sano :
アザビシクロブタンを活用するキノロン系抗菌剤の合成開発,
日本薬学会第125年会, Mar. 2005.
70. Yoshimitsu Nagao, 谷本 典昭, 本城 崇 and Shigeki Sano :
プロキラルな環状カルボン酸無水物の触媒的不斉チオリシス,
日本薬学会第125年会, Mar. 2005.
71. Yoshimitsu Nagao, 陳 青根 and Shigeki Sano :
アルキニルフルオロシランの合成法の開発と応用研究,
日本薬学会第125年会, Mar. 2005.
72. Yoshimitsu Nagao, 宮本 素行, 三谷 智子 and Shigeki Sano :
MgBr2触媒を活用するDarzens反応の開発,
日本薬学会第125年会, Mar. 2005.
73. Yoshimitsu Nagao, 本城 崇 and Shigeki Sano :
新規含硫黄有機触媒を用いた環状酸無水物のエナンチオ選択的チオリシス,
日本薬学会第125年会, Mar. 2005.
74. Yoshimitsu Nagao, Tinh Van Dang, 宮本 素行 and Shigeki Sano :
キラルなcAMP-特異的ホスホジエステラーゼ阻害剤の実用的合成,
日本薬学会第125年会, Mar. 2005.
75. Yoshimitsu Nagao, 林 一彦, 小川 志穂 and Shigeki Sano :
含イオウ常用医薬品に関する情報収集,
日本薬学会第125年会, Mar. 2005.
76. Shigeki Sano, 黒田 陽子 and Yoshimitsu Nagao :
フルオロオレフィンを基盤とする新規ジペプチドミメティクス合成法の開発研究,
日本薬学会第125年会, Mar. 2005.
77. Shigeki Sano, 原田 悦子 and Yoshimitsu Nagao :
二重結合の転位を基盤とするβ,γ-不飽和エステルの合成,
日本薬学会第125年会, Mar. 2005.
78. Shigeki Sano, Michiyasu Nakao and Yoshimitsu Nagao :
酵素アセチル化反応を用いるα-メチルセリン誘導体のエナンチオ分岐的合成,
日本薬学会第125年会, Mar. 2005.
79. Shigeki Sano, 久次米 永子 and Yoshimitsu Nagao :
新規ホスホノ酢酸エステルの合成と不斉HWE反応への応用,
日本薬学会第125年会, Mar. 2005.
80. Shigeki Sano, 安部 忍 and Yoshimitsu Nagao :
イソマンニド誘導体をキラル補助基とする不斉HWE反応,
日本薬学会第125年会, Mar. 2005.
81. Yoshimitsu Nagao, 池江 克文, 中島 正晃, 林 一彦 and Shigeki Sano :
1-アザビシクロ[1.1.0]ブタンから誘導したアゼチジン誘導体を活用する新規キノロン系抗菌剤の合成開発研究,
第34回複素環化学討論会, Nov. 2004.
82. Yoshimitsu Nagao, 熊沢 益徳, 田中 悟 and Shigeki Sano :
新規なフラン環合成法の開発研究,
第34回複素環化学討論会, Nov. 2004.
83. 谷本 典昭, 本城 崇, Shigeki Sano and Yoshimitsu Nagao :
プロキラルな環状カルボン酸無水物の触媒的不斉チオリシス,
第43回日本薬学会·日本病院薬剤師会中国四国支部学術大会, Nov. 2004.
84. Shigeki Sano, 黒田 陽子 and Yoshimitsu Nagao :
フルオロオレフィンイソステアを基盤とするペプチドミメティクス合成,
第43回日本薬学会·日本病院薬剤師会中国四国支部学術大会, Nov. 2004.
85. Shigeki Sano, 原田 悦子 and Yoshimitsu Nagao :
α,β-不飽和カルボン酸のタンデム型二重結合転位-エステル化反応,
第43回日本薬学会·日本病院薬剤師会中国四国支部学術大会, Nov. 2004.
86. Shigeki Sano, Michiyasu Nakao and Yoshimitsu Nagao :
酵素反応を用いるα-メチルセリン誘導体のエナンチオ分岐的合成,
第43回日本薬学会·日本病院薬剤師会中国四国支部学術大会, Nov. 2004.
87. Shigeki Sano, 久次米 永子 and Yoshimitsu Nagao :
キラルなリン原子を有する新規ホスホノ酢酸エステルの合成,
第43回日本薬学会·日本病院薬剤師会中国四国支部学術大会, Nov. 2004.
88. Shigeki Sano, 安部 忍 and Yoshimitsu Nagao :
α-メチルホスホノ酢酸エステルの不斉HWE反応,
第43回日本薬学会·日本病院薬剤師会中国四国支部学術大会, Nov. 2004.
89. Yoshimitsu Nagao, 林 一彦, 中島 正晃, 池江 克文, Shigeki Sano, 佐藤 千里, 磯田 武寿, 玉井 聖, 阿部 隆夫 and 熊谷 年夫 :
高歪み分子1-Azabicyclo[1.1.0]butaneの合成と新規抗菌剤合成への応用,
第30回反応と合成の進歩シンポジウム, Oct. 2004.
90. Yoshimitsu Nagao, 熊沢 益徳, 田中 悟 and Shigeki Sano :
環状ヒドロキシ共役エノン体のシリカゲルを用いた環拡大反応の開発,
日本薬学会第124年会, Mar. 2004.
91. Yoshimitsu Nagao, 宮本 素行 and Shigeki Sano :
α-ハロケトンを用いるアルドール反応及びその不斉反応への応用,
日本薬学会第124年会, Mar. 2004.
92. Yoshimitsu Nagao, 本城 崇 and Shigeki Sano :
環状酸無水物の効率的モノアルキル化反応の開発研究,
日本薬学会第124年会, Mar. 2004.
93. Shigeki Sano, 中野 文仁, 竹本 裕香, 久次米 永子 and Yoshimitsu Nagao :
新規光学活性ホスホノ酢酸エステルを用いるエナンチオ選択的HWE反応,
日本薬学会第124年会, Mar. 2004.
94. Shigeki Sano, 竹本 裕香, 久次米 永子, 中野 文仁 and Yoshimitsu Nagao :
キラルなリン原子を有する新規HWE試薬の合成,
日本薬学会第124年会, Mar. 2004.
95. Shigeki Sano, 畦津 知宏, 中野 文仁 and Yoshimitsu Nagao :
タンデム型二重結合転位-エステル化反応によるβ,γ-不飽和エステルの合成,
日本薬学会第124年会, Mar. 2004.
96. Shigeki Sano, 中野 文仁, 竹本 裕香, 久次米 永子 and Yoshimitsu Nagao :
2-置換-1,3-ジオキサン-5-オンを基質とするHWE反応,
第42回日本薬学会·日本病院薬剤師会中国四国支部学術大会, Nov. 2003.
97. Shigeki Sano, 竹本 裕香, 久次米 永子, 中野 文仁 and Yoshimitsu Nagao :
キラルなリン原子を有する新しいHWE試薬,
第42回日本薬学会·日本病院薬剤師会中国四国支部学術大会, Nov. 2003.
98. Shigeki Sano, 畦津 知宏, 東雲 三和 and Yoshimitsu Nagao :
転位-エステル化反応によるβ,γ-不飽和エステルの合成,
第42回日本薬学会·日本病院薬剤師会中国四国支部学術大会, Nov. 2003.
99. Shigeki Sano, 竹本 裕香, 久次米 永子, 中野 文仁 and Yoshimitsu Nagao :
ホスホノ酢酸ジアニオンを用いる立体選択的HWE反応,
第33回複素環化学討論会, Oct. 2003.
100. Yoshimitsu Nagao, 本城 崇, 飯森 均, Satoru GOTO, Shigeki Sano and 城 始勇 :
分子内非結合性相互作用を有するチアゾール及びオキサゾール誘導体の分子構造特性,
第33回複素環化学討論会, Oct. 2003.
101. Yoshimitsu Nagao, 宮本 素行, 宮本 聡 and Shigeki Sano :
アキラル及びキラルなピロリドン誘導体を活用する不斉Pummerer反応及び不斉Aldol反応,
第33回複素環化学討論会, Oct. 2003.
102. Yoshimitsu Nagao, 宮本 素行, 柏木 貴雄 and Shigeki Sano :
立体選択的不斉Pummerer反応及びPummerer型環化反応の検討,
日本薬学会第123年会, Mar. 2003.
103. Yoshimitsu Nagao, 田中 悟, 植木 章晴, 熊沢 益徳, Shigeki Sano and 城 始勇 :
環状ヒドロキシ共役エノン体のPd(0)触媒環拡大反応の開発,
日本薬学会第123年会, Mar. 2003.
104. Yoshimitsu Nagao, 田中 悟, 植木 章晴, 浅野 和徳, 熊沢 益徳 and Shigeki Sano :
Pd(II)触媒-DDQを用いた3-Alkylidene Isoindolinone誘導体の合成開発,
日本薬学会第123年会, Mar. 2003.
105. Yoshimitsu Nagao, 木村 めぐみ, 小倉 佑樹 and Shigeki Sano :
抗緑膿菌活性を有するN-アリールイソチアゾロン誘導体の合成研究,
日本薬学会第123年会, Mar. 2003.
106. Shigeki Sano, 中野 文仁 and Yoshimitsu Nagao :
キラルアミノアルコールを不斉源とするエナンチオ選択的HWE反応,
日本薬学会第123年会, Mar. 2003.
107. Shigeki Sano, 竹本 裕香 and Yoshimitsu Nagao :
アリールアルキルケトンを基質とするE選択的HWE反応,
日本薬学会第123年会, Mar. 2003.
108. Shigeki Sano, 畦津 知宏, 中野 文仁 and Yoshimitsu Nagao :
イソマンニドおよびイソソルビド誘導体を不斉補助基とするジアステレオ選択的HWE反応,
日本薬学会第123年会, Mar. 2003.
109. Yoshimitsu Nagao, 本城 崇, 飯盛 均, Satoru GOTO, Shigeki Sano and 城 始勇 :
分子内非結合性相互作用を有するチアゾール誘導体の合成及び分子構造特性,
日本薬学会第123年会, Mar. 2003.
110. Yoshimitsu Nagao, 本城 崇, Satoru GOTO, 飯森 均, Shigeki Sano and 城 始勇 :
分子内非結合性相互作用を有するチアジアゾール及びチアゾール誘導体の分子構造特性と機能性,
第32回複素環化学討論会, Dec. 2002.
111. Shigeki Sano, 中野 文仁 and Yoshimitsu Nagao :
プロキラルケトンを基質とするエナンチオ選択的不斉HWE反応,
第41回日本薬学会·日本病院薬剤師会中国四国支部学術大会, Nov. 2002.
112. Shigeki Sano, 竹本 裕香 and Yoshimitsu Nagao :
ホスホノ酢酸ジアニオンとアリールアルキルケトンのE選択的HWE反応,
第41回日本薬学会·日本病院薬剤師会中国四国支部学術大会, Nov. 2002.
113. Shigeki Sano, 畦津 知宏, 中野 文仁 and Yoshimitsu Nagao :
イソマンニドおよびイソソルビド誘導体をキラル補助基とする不斉HWE反応,
第41回日本薬学会·日本病院薬剤師会中国四国支部学術大会, Nov. 2002.
114. Yoshimitsu Nagao, 飯盛 均, 本城 崇, Hiroshi Chuman, Satoru GOTO, Shigeki Sano and 城 始勇 :
分子内非結合性S---Halogen (F, Cl, Br) 相互作用を有する新規複素環化合物の合成; 構造特性及び抗腫瘍活性,
日本薬学会第122年会, Mar. 2002.
115. Yoshimitsu Nagao, 飯盛 均, 前田 知子, Hiroshi Chuman, Satoru GOTO, Shigeki Sano and 城 始勇 :
分子内非結合性相互作用を有する新規複素環化合物の合成; 構造特性及び反応性,
日本薬学会第121年会, Mar. 2001.
116. Yoshimitsu Nagao, 飯森 均, Hiroshi Chuman, Satoru GOTO, 平田 晃陰, Shigeki Sano and 城 始勇 :
非結合性S---X (X＝O, S) 相互作用を有する新規有機硫黄化合物の合成とその構造特性,
第39回日本薬学会·日本病院薬剤師会中国四国支部学術大会, Oct. 2000.
117. Yoshimitsu Nagao, 飯森 均, Satoru GOTO, Hiroshi Chuman, Shigeki Sano and 城 始勇 :
分子内非結合性相互作用が期待される有機硫黄化合物の合成と構造特性,
第18回有機合成化学夏期大学, Aug. 2000.
118. Yoshimitsu Nagao, 飯森 均, Hiroshi Chuman, Satoru GOTO, 平田 晃陰, Shigeki Sano and 城 始勇 :
非結合性相互作用を基盤とする回転; 幾何; 互変異性体が可能な複素環化合物の優先構造,
日本薬学会第120年会, Mar. 2000.
119. Yoshimitsu Nagao, 飯森 均, Satoru GOTO, 平田 晃陰, Shigeki Sano and Hiroshi Chuman :
非結合性S---X (X=S,O,Br,π) 相互作用が期待される新規複素環化合物の合成とその構造特性,
第26回ヘテロ原子化学討論会, Dec. 1999.
120. Yoshimitsu Nagao, 飯森 均, 平田 晃陰, Satoru GOTO, Shigeki Sano and 城 始勇 :
分子内及び分子間非結合性S---X (X＝O, N, S, etc.) 相互作用が期待される新規有機硫黄化合物の合成,
日本薬学会119年会, Mar. 1999.
121. Yoshimitsu Nagao, 飯森 均, Satoru GOTO, 平田 晃陰, 西島 宏明, 後河内 秀樹, Shigeki Sano and 城 始勇 :
非結合性S---X (X＝O, S, N) 相互作用を有する有機硫黄化合物の合成とその証明,
第24回反応と合成の進歩シンポジウム, Oct. 1998.
122. 平田 晃陰, Satoru GOTO, Shigeki Sano, Yoshimitsu Nagao and 城 始勇 :
Angiotensin II受容体拮抗作用を示すAcyliminothiadiazoline誘導体の特異な物性と構造活性相関,
第25回構造活性相関シンポジウム, Nov. 1997.
123. Yoshimitsu Nagao, 平田 晃陰, Satoru GOTO, Shigeki Sano and 城 始勇 :
創薬デザインの新展開: S---O非結合性相互作用の重要性,
日本薬学会第117年会, Mar. 1997.
124. 平田 晃陰, 奥平 正泰, Satoru GOTO and Yoshimitsu Nagao :
Angiotensin II受容体拮抗作用を有するAcyliminothiadiazoline誘導体の定量的構造活性相関,
第5回日本薬学会医薬化学部会年会, Oct. 1996.

Report:

1. Yoshimitsu Nagao and Shigeki Sano :
平成16年度∼平成18年度科学研究費補助金(基盤研究(B))研究成果報告書,
May 2007.
2. Yoshimitsu Nagao and Shigeki Sano :
平成14年度∼平成15年度科学研究費補助金(基盤研究(B)(2))研究成果報告書,
May 2004.
3. Yoshimitsu Nagao and Shigeki Sano :
平成12年度∼平成13年度科学研究費補助金(基盤研究(B)(2))研究成果報告書,
Mar. 2002.
4. Yoshimitsu Nagao and Shigeki Sano :
平成10年度∼平成11年度科学研究費補助金(基盤研究(B)(2))研究成果報告書,
Mar. 2000.
5. Yoshimitsu Nagao and Shigeki Sano :
平成8年度∼平成9年度科学研究費補助金(基盤研究(B)(2))研究成果報告書,
Mar. 1998.

Patent:

1. Yoshimitsu Nagao and Shigeki Sano : セリン誘導体の製造方法, 09-088620 (Mar. 1997), .
2. Yoshimitsu Nagao and Shigeki Sano : 新規γ-ラクトン誘導体, 04-260584 (Sep. 1992), .
3. Yoshimitsu Nagao and Shigeki Sano : 新規ピロリジン誘導体又はその塩を有効成分とする抗腫瘍剤，及びポリヒドロキシ化高級脂肪酸置換ピロリジン誘導体, 04-260585 (Sep. 1992), .
4. Yoshimitsu Nagao and Shigeki Sano : トリアゾール誘導体, 03-017067 (Jan. 1991), .

Grants-in-Aid for Scientific Research (KAKEN Grants Database @ NII.ac.jp)

  • イオウ原子の非結合性相互作用を機軸とする斬新な創薬メソドロジーの構築 (Project/Area Number: 16659030 )
  • Development of Synthetic Methods for the Silaallene Cationic Species and the Related Compounds and Their Application Reactions (Project/Area Number: 16390008 )
  • 赤外線蛍光内視鏡診断のための赤外蛍光増強剤の開発 (Project/Area Number: 15659173 )
  • Molecular Design, Syntheses, and Utilization of New Thiazole-Related Compounds (Project/Area Number: 14370723 )
  • 二箇所同一不斉認識場を有するキラルビスチアゾリン誘導体を活用する不斉誘導反応 (Project/Area Number: 14044075 )
  • 高感度赤外線蛍光内視鏡を用いた微小癌診断法の開発 (Project/Area Number: 13218088 )
  • 各種アレン置換基を有する複素環化合物のパラジウム触媒環拡大反応 (Project/Area Number: 13029085 )
  • 天然アミノ酸を素材とした不斉加水分解能を有する人工酵素のデザイン合成開発 (Project/Area Number: 12877350 )
  • Construction of New Reaction Media and Its Application Based on the Non-bonded Interaction Concept (Project/Area Number: 12470482 )
  • 赤外線蛍光内視鏡を用いた微小癌診断法の開発 (Project/Area Number: 12217100 )
  • 硫黄原子を基盤とする非結合性相互作用の解明と新機能性分子の合成開発 (Project/Area Number: 11120239 )
  • Synthesis and Characterization of New Functional Molecules Involving the Nonbonded Sulfur-Heteroatom Interactions (Project/Area Number: 10470470 )
  • 非結合性相互作用を有する新規分子の合成とその医薬品リード化合物開発への応用 (Project/Area Number: 10169247 )
  • 芳香環ラジカル求核置換反応(S_<RN>Ar)を基盤とする不斉環化反応の開発 (Project/Area Number: 10125228 )
  • 生体模倣反応や特異物性を分子設計の基盤とするカテプシン類阻害剤の合成開発 (Project/Area Number: 09273244 )
  • カスケード反応を基盤とする新規生物活性複素環の構築 (Project/Area Number: 09231235 )
  • Studies on the Development of New Reaction Modes for the Synthesis of New Drugs (Project/Area Number: 08457585 )
  • 潜在的活性種を活用する実践的環化反応の開発研究 (Project/Area Number: 08245238 )
  • ルイス酸-アレニルケトン系を利用する新規な不斉環化反応の開発 (Project/Area Number: 07214223 )
  • Development of New Cysteine Proteinase Inhibitors Involving the Generation of Conjugated Allenyl Esters as the Latent Active Species (Project/Area Number: 06453215 )
  • DEVELOPMENTAL RESEARCH TO UTILIZE MICROORGANISM PRODUCTS HAVING POTENCY OF BIOFUNCTIONAL CONTROL FOR DRUG MATERIALS (Project/Area Number: 06303014 )
  • 化学選択的反応を基盤とする高選択的不斉分岐反応 (Project/Area Number: 06225225 )
  • 抗癌剤開発を志向する新規なポリオキシ高級脂肪酸エステルの合成研究 (Project/Area Number: 04152085 )
  • 新規構造を有する天然物由来抗癌物質に関する研究 (Project/Area Number: 04151016 )
  • 新規構造を有する天然物由来抗癌物質に関する研究 (Project/Area Number: 03151016 )
  • Design of the Molecules Bearing Specific Stereochemistry and Its Application to the Development of New Reactions (Project/Area Number: 02453141 )
  • 天然物由来制癌物質の探索とその化学的誘導に関する研究 (Project/Area Number: 02151018 )
  • 特定酵素に高選択的な分子認識並びに反応性を示す抗癌剤の合成開発研究 (Project/Area Number: 01015053 )
  • 天然物由来制癌物質の探索とその化学的誘導に関する研究 (Project/Area Number: 01010018 )
  • Construction of Chiral Building Blocks through Enantioselective Protonation (Project/Area Number: 63430024 )
  • 放射線の制がん効果を増強する薬剤の開発とスクリーニングシステムの確立に関する研究 (Project/Area Number: 63010069 )
  • ハイパーバレント有機スズ化合物による反応の立体制御と抗癌剤の開発研究 (Project/Area Number: 62570938 )
  • Carbene-Type Reactive Intermediates: Novel Physical Properties and Synthetic Applications (Project/Area Number: 62300014 )
  • 放射線の制がん効果を増強する薬剤の開発とスクリーニングシステムの確立に関する研究 (Project/Area Number: 62010070 )
  • 放射線の制がん効果を増強する薬剤の開発とスクリーニングシステムの確立に関する研究 (Project/Area Number: 61010070 )
  • Design and Synthetic Development of New Multifunctional Anti-cancer Agents (Project/Area Number: 60470146 )
  • Search by Researcher Number (40027074)